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Literature summary for 3.4.21.35 extracted from

  • Oliva, M.L.; Mendes, C.R.; Juliano, M.A.; Chagas, J.R.; Rosa, J.C.; Greene, L.J.; Sampaio, M.U.; Sampaio, C.A.
    Characterization of a tissue kallikrein inhibitor isolated from Bauhinia bauhinioides seeds: inhibition of the hydrolysis of kininogen related substrates (1999), Immunopharmacology, 45, 163-169.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
Bauhinia bauhinioides trypsin inhibitor II i.e. BbTI-II; N-terminal sequence of the protein is SVVVDTNGQPVSNGADAYYLV Sus scrofa
additional information no inhibition by Bauhinia bauhinioides trypsin inhibitor I Homo sapiens
additional information no inhibition by Bauhinia bauhinioides trypsin inhibitor I Sus scrofa

Localization

Localization Comment Organism GeneOntology No. Textmining
extracellular secretion Homo sapiens
-
-

Natural Substrates/ Products (Substrates)

Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
polypeptide + H2O Homo sapiens
-
peptides
-
?
polypeptide + H2O Sus scrofa
-
peptides
-
?

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
-
-
Sus scrofa
-
commercial product
-

Source Tissue

Source Tissue Comment Organism Textmining
pancreas
-
Homo sapiens
-
pancreas
-
Sus scrofa
-
urine
-
Homo sapiens
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
polypeptide + H2O
-
Homo sapiens peptides
-
?
polypeptide + H2O
-
Sus scrofa peptides
-
?
Pro-Phe-Arg-7-amido-4-methylcoumarin + H2O
-
Homo sapiens Pro-Phe-Arg + 7-amino-4-methylcoumarin
-
?
Pro-Phe-Arg-7-amido-4-methylcoumarin + H2O
-
Sus scrofa Pro-Phe-Arg + 7-amino-4-methylcoumarin
-
?

Temperature Optimum [°C]

Temperature Optimum [°C] Temperature Optimum Maximum [°C] Comment Organism
37
-
assay at Homo sapiens
37
-
assay at Sus scrofa

pH Optimum

pH Optimum Minimum pH Optimum Maximum Comment Organism
8
-
assay at Homo sapiens
8
-
assay at Sus scrofa

Ki Value [mM]

Ki Value [mM] Ki Value maximum [mM] Inhibitor Comment Organism Structure
0.000002
-
Bauhinia bauhinioides trypsin inhibitor II pH 8.0, 37°C Sus scrofa