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Literature summary for 3.4.21.21 extracted from

  • Stone, M.D.; Harvey, S.B.; Martinez, M.B.; Bach, R.R.; Nelsestuen, G.L.
    Large enhancement of functional activity of active site-inhibited factor VIIa due to protein dimerization: insights into mechanism of assembly/disassembly from tissue factor (2005), Biochemistry, 44, 6321-6330.
    View publication on PubMed

Activating Compound

Activating Compound Comment Organism Structure
tissue factor
-
Homo sapiens

Inhibitors

Inhibitors Comment Organism Structure
dimeric active site-inhibited blood clotting factor VIIa dimeric fVIIai, 16000fold inhibitory effect Homo sapiens

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
-
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
D-isoleucyl-L-prolyl-L-arginine-p-nitroanilide + H2O
-
Homo sapiens D-isoleucyl-L-prolyl-L-arginine + p-nitroaniline
-
?
D-phenylalanyl-L-pipecolyl-L-arginine-p-nitroanilide + H2O
-
Homo sapiens D-phenylalanyl-L-pipecolyl-L-arginine + p-nitroaniline
-
?
factor X + H2O
-
Homo sapiens factor Xa
-
?
Z-D-arginyl-glycyl-arginine-p-nitroanilide + H2O
-
Homo sapiens Z-D-arginyl-glycyl-arginine + p-nitroaniline
-
?

Synonyms

Synonyms Comment Organism
factor VIIa
-
Homo sapiens
FVIIa
-
Homo sapiens