Inhibitors | Comment | Organism | Structure |
---|---|---|---|
1-(2,4-dichlorobenzoyl)-N-methyl-1H-indazole-3-carboxamide | - |
Homo sapiens | |
2-(3-(2-hydroxyethyl)ureido)-N-(2-methoxybenzyl)-1H-benzo[d]imidazole-5-sulfonamide | - |
Homo sapiens | |
2-(3-(2-hydroxyethyl)ureido)-N-(2-methylbenzyl)-1H-benzo[d]imidazole-5-sulfonamide | - |
Homo sapiens | |
2-{[(2-hydroxyethyl)carbamoyl]amino}-N-[(2-methoxyphenyl)methyl]-1H-benzimidazole-5-sulfonamide | - |
Homo sapiens | |
DV-1006 | - |
Homo sapiens | |
ethyl 1-(2,4-dichlorobenzoyl)-1H-indazole-3-carboxylate | - |
Homo sapiens | |
KF950 | - |
Homo sapiens | |
N,N-bis(2-hydroxyethyl)-5-(4-methoxyphenyl)-1H-pyrazole-3-carboxamide | - |
Homo sapiens | |
N-(2-chlorobenzyl)-2-(3-(2-hydroxyethyl)ureido)-1H-benzo[d]imidazole-5-sulfonamide | - |
Homo sapiens | |
N-(2-fluorobenzyl)-2-(3-(2-hydroxyethyl)ureido)-1H-benzo[d]imidazole-5-sulfonamide | - |
Homo sapiens | |
N-(2-hydroxyethyl)-5-(4-methoxyphenyl)-N-methyl-1H-pyrazole-3-carboxamide | - |
Homo sapiens | |
N-(2-hydroxypropyl)-5-(4-methoxyphenyl)-1H-pyrazole-3-carboxamide | - |
Homo sapiens | |
N-(3, 5-difluorobenzyl)-2-(3-(2-hydroxyethyl)ureido)-1H-benzo[d]imidazole-5-sulfonamide | - |
Homo sapiens | |
N-(3,5-dichlorobenzyl)-2-(3-(2-hydroxyethyl)ureido)-1H-benzo[d]imidazole-5-sulfonamide | - |
Homo sapiens | |
N-(3-hydroxypropyl)-5-(4-methoxyphenyl)-1H-pyrazole-3-carboxamide | - |
Homo sapiens | |
N-(5-bromobenzo[d]thiazol-2-yl)-2-(4-pentylpiperazin-1-yl)acetamide | - |
Homo sapiens | |
N-(5-bromobenzo[d]thiazol-2-yl)-2-(diisopentylamino)acetamide | - |
Homo sapiens | |
N-(5-bromobenzo[d]thiazol-2-yl)-2-(dipentylamino)acetamide | - |
Homo sapiens | |
N-(6-bromobenzo[d]thiazol-2-yl)-2-(dibutylamino)acetamide | - |
Homo sapiens | |
N-alpha-tosyl-L-lysyl-chloromethyl-ketone | - |
Homo sapiens | |
N-benzyl-2-(3-(2-hydroxyethyl)ureido)-1H-benzo[d]imidazole-5-sulfonamide | - |
Homo sapiens | |
N-hexyl-2-(3-(2-hydroxyethyl)ureido)-1H-benzo[d]imidazole-5-sulfonamide | - |
Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
- |
- |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
0.08 | - |
pH and temperature not specified in the publication | Homo sapiens | N-(2-fluorobenzyl)-2-(3-(2-hydroxyethyl)ureido)-1H-benzo[d]imidazole-5-sulfonamide | |
0.28 | - |
pH and temperature not specified in the publication | Homo sapiens | N-benzyl-2-(3-(2-hydroxyethyl)ureido)-1H-benzo[d]imidazole-5-sulfonamide | |
0.34 | - |
pH and temperature not specified in the publication | Homo sapiens | N-(3, 5-difluorobenzyl)-2-(3-(2-hydroxyethyl)ureido)-1H-benzo[d]imidazole-5-sulfonamide | |
0.54 | - |
pH and temperature not specified in the publication | Homo sapiens | N-(5-bromobenzo[d]thiazol-2-yl)-2-(dipentylamino)acetamide | |
1.06 | - |
pH and temperature not specified in the publication | Homo sapiens | N-(2-chlorobenzyl)-2-(3-(2-hydroxyethyl)ureido)-1H-benzo[d]imidazole-5-sulfonamide | |
1.09 | - |
pH and temperature not specified in the publication | Homo sapiens | N-(5-bromobenzo[d]thiazol-2-yl)-2-(diisopentylamino)acetamide | |
1.43 | - |
pH and temperature not specified in the publication | Homo sapiens | N-(3-hydroxypropyl)-5-(4-methoxyphenyl)-1H-pyrazole-3-carboxamide | |
1.62 | - |
pH and temperature not specified in the publication | Homo sapiens | N-hexyl-2-(3-(2-hydroxyethyl)ureido)-1H-benzo[d]imidazole-5-sulfonamide | |
2.45 | - |
pH and temperature not specified in the publication | Homo sapiens | N-(3,5-dichlorobenzyl)-2-(3-(2-hydroxyethyl)ureido)-1H-benzo[d]imidazole-5-sulfonamide | |
2.78 | - |
pH and temperature not specified in the publication | Homo sapiens | N-(6-bromobenzo[d]thiazol-2-yl)-2-(dibutylamino)acetamide | |
3.24 | - |
pH and temperature not specified in the publication | Homo sapiens | ethyl 1-(2,4-dichlorobenzoyl)-1H-indazole-3-carboxylate | |
3.78 | - |
pH and temperature not specified in the publication | Homo sapiens | 1-(2,4-dichlorobenzoyl)-N-methyl-1H-indazole-3-carboxamide | |
5.08 | - |
pH and temperature not specified in the publication | Homo sapiens | N-(5-bromobenzo[d]thiazol-2-yl)-2-(4-pentylpiperazin-1-yl)acetamide | |
5.45 | - |
pH and temperature not specified in the publication | Homo sapiens | 2-(3-(2-hydroxyethyl)ureido)-N-(2-methylbenzyl)-1H-benzo[d]imidazole-5-sulfonamide | |
5.73 | - |
pH and temperature not specified in the publication | Homo sapiens | N,N-bis(2-hydroxyethyl)-5-(4-methoxyphenyl)-1H-pyrazole-3-carboxamide | |
6.04 | - |
pH and temperature not specified in the publication | Homo sapiens | 2-(3-(2-hydroxyethyl)ureido)-N-(2-methoxybenzyl)-1H-benzo[d]imidazole-5-sulfonamide | |
6.81 | - |
pH and temperature not specified in the publication | Homo sapiens | N-(2-hydroxyethyl)-5-(4-methoxyphenyl)-N-methyl-1H-pyrazole-3-carboxamide | |
7.32 | - |
pH and temperature not specified in the publication | Homo sapiens | 2-{[(2-hydroxyethyl)carbamoyl]amino}-N-[(2-methoxyphenyl)methyl]-1H-benzimidazole-5-sulfonamide | |
8.92 | - |
pH and temperature not specified in the publication | Homo sapiens | N-(2-hydroxypropyl)-5-(4-methoxyphenyl)-1H-pyrazole-3-carboxamide | |
142.6 | - |
pH and temperature not specified in the publication | Homo sapiens | N-alpha-tosyl-L-lysyl-chloromethyl-ketone |