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Literature summary for 3.4.14.5 extracted from

  • Reinhold, D.; Goihl, A.; Wrenger, S.; Reinhold, A.; Kuehlmann, U.C.; Faust, J.; Neubert, K.; Thielitz, A.; Brocke, S.; Taeger, M.; Ansorge, S.; Bank, U.
    Role of dipeptidyl peptidase IV (DP IV)-like enzymes in T lymphocyte activation: investigations in DP IV/CD26-knockout mice (2009), Clin. Chem. Lab. Med., 47, 268-274.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
DP IV-I3 selective DP IV inhibitor, 87% inhibition at 0.01 mM Mus musculus
Lys[Z(NO2)]-pyrrolidide non-selective inhibitor of DP IV-like activity; non-specific DPIV inhibitor, 96% inhibition at 0.01 mM Mus musculus
Lys[Z(NO2)]-thiazolidide non-selective inhibitor of DP IV-like activity; non-specific DPIV inhibitor Mus musculus
[(2R)-4-oxo-4-[3-(trifluoromethyl)-5,6-dihydro-1,2,4[triazolo]4,3-alpha]pyrazin-7(8H)-yl]-1-(2,5-difluorophenyl)butan-2-amine hydrochloride selective DP IV inhibitor Mus musculus

Organism

Organism UniProt Comment Textmining
Mus musculus
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
spleen
-
Mus musculus
-
splenocyte
-
Mus musculus
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
Gly-Pro-7-amido-4-methylcoumarin + H2O
-
Mus musculus Gly-Pro + 7-amino-4-methylcoumarin
-
?

Synonyms

Synonyms Comment Organism
CD26
-
Mus musculus
dipeptidyl peptidase IV
-
Mus musculus
DP IV
-
Mus musculus

General Information

General Information Comment Organism
physiological function dipeptidyl peptidase IV regulates T lymphocyte activation Mus musculus