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Literature summary for 3.4.14.5 extracted from

  • Gilmore, B.F.; Carson, L.; McShane, L.L.; Quinn, D.; Coulter, W.A.; Walker, B.
    Synthesis, kinetic evaluation, and utilization of a biotinylated dipeptide proline diphenyl phosphonate for the disclosure of dipeptidyl peptidase IV-like serine proteases (2006), Biochem. Biophys. Res. Commun., 347, 373-379.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
diphenyl [1-(N-(15-oxo-19-[(4R)-2-oxohexahydro-1H-thieno[3,4-d]imidazol-4-yl]-4,7,10-trioxa-14-azanonadec-1-yl)-L-glutaminyl)pyrrolidin-2-yl]phosphonate irreversible inhibitor Sus scrofa

Organism

Organism UniProt Comment Textmining
Sus scrofa
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
kidney
-
Sus scrofa
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
Gly-Pro-4-methylcoumarin 7-amide + H2O
-
Sus scrofa Gly-Pro + 7-amino-4-methylcoumarin
-
?

Ki Value [mM]

Ki Value [mM] Ki Value maximum [mM] Inhibitor Comment Organism Structure
0.04316
-
diphenyl [1-(N-(15-oxo-19-[(4R)-2-oxohexahydro-1H-thieno[3,4-d]imidazol-4-yl]-4,7,10-trioxa-14-azanonadec-1-yl)-L-glutaminyl)pyrrolidin-2-yl]phosphonate
-
Sus scrofa