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Literature summary for 3.1.3.5 extracted from

  • Li, R.W.; Man, R.Y.; Vanhoutte, P.M.; Leung, G.P.
    Stimulation of ecto-5'-nucleotidase in human umbilical vein endothelial cells by lipopolysaccharide (2008), Am. J. Physiol. Heart Circ. Physiol., 295, H1177-H1181.
    View publication on PubMed

Activating Compound

Activating Compound Comment Organism Structure
ammonium pyrrolidin dithiocarbamate 0.01 mM ammonium pyrrolidin dithiocarbamate increases the basal activity of ecto-5'-nucleotidase by 17% but has no effect on the lipopolysaccharide-induced increase in ecto-5'-nucleotidase activity Homo sapiens
lipopolysaccharide ecto-5'-nucleotidase activity increases after incubation with 10 ng/ml lipopolysaccharide for 24 h but is not changed after shorter incubation times Homo sapiens

Inhibitors

Inhibitors Comment Organism Structure
adenosine 5'-(alpha,beta-methylene)diphosphate complete inhibition at 0.1 mM Homo sapiens
Ly-294002 0.01 mM LY-294002 abolishes lipopolysaccharide-induced ecto-5'-nucleotidase activity Homo sapiens

Localization

Localization Comment Organism GeneOntology No. Textmining
membrane
-
Homo sapiens 16020
-

Molecular Weight [Da]

Molecular Weight [Da] Molecular Weight Maximum [Da] Comment Organism
70000
-
SDS-PAGE Homo sapiens

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
-
-

Posttranslational Modification

Posttranslational Modification Comment Organism
glycoprotein
-
Homo sapiens

Source Tissue

Source Tissue Comment Organism Textmining
HUVEC cell
-
Homo sapiens
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
5'-AMP + H2O
-
Homo sapiens adenosine + phosphate
-
?

Synonyms

Synonyms Comment Organism
CD73
-
Homo sapiens
E-5'-Nu
-
Homo sapiens
ecto-5'-nucleotidase
-
Homo sapiens