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Literature summary for 2.7.11.26 extracted from

  • Llorach-Pares, L.; Nonell-Canals, A.; Avila, C.; Sanchez-Martinez, M.
    Kororamides, convolutamines, and indole derivatives as possible tau and dual-specificity kinase inhibitors for Alzheimer's disease A computational study (2018), Mar. Drugs, 16, 386 .
    View publication on PubMedView publication on EuropePMC
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Inhibitors

Inhibitors Comment Organism Structure
(5,6-dibromo-1H-indol-3-yl)methanol
-
 Homo sapiens
(5,6-dichloro-1H-indol-3-yl)methanol
-
 Homo sapiens
(5,6-difluoro-1H-indol-3-yl)methanol
-
 Homo sapiens
(5-bromo-6-chloro-1H-indol-3-yl)methanol
-
 Homo sapiens
(5-bromo-6-fluoro-1H-indol-3-yl)methanol
-
 Homo sapiens
(6-bromo-5-chloro-1H-indol-3-yl)methanol
-
 Homo sapiens
(6-bromo-5-fluoro-1H-indol-3-yl)methanol
-
 Homo sapiens
1-(5,6-dibromo-1H-indol-3-yl)methanamine
-
 Homo sapiens
1-(5,6-dibromo-1H-indol-3-yl)propan-2-one
-
 Homo sapiens
1-(5,6-dichloro-1H-indol-3-yl)methanamine
-
 Homo sapiens
1-(5,6-dichloro-1H-indol-3-yl)propan-2-one
-
 Homo sapiens
1-(5,6-difluoro-1H-indol-3-yl)methanamine
-
 Homo sapiens
1-(5,6-difluoro-1H-indol-3-yl)propan-2-one
-
 Homo sapiens
1-(5-bromo-6-chloro-1H-indol-3-yl)methanamine
-
 Homo sapiens
1-(5-bromo-6-chloro-1H-indol-3-yl)propan-2-one
-
 Homo sapiens
1-(5-bromo-6-fluoro-1H-indol-3-yl)methanamine
-
 Homo sapiens
1-(5-bromo-6-fluoro-1H-indol-3-yl)propan-2-one
-
 Homo sapiens
1-(6-bromo-5-chloro-1H-indol-3-yl)methanamine
-
 Homo sapiens
1-(6-bromo-5-chloro-1H-indol-3-yl)propan-2-one
-
 Homo sapiens
1-(6-bromo-5-fluoro-1H-indol-3-yl)methanamine
-
 Homo sapiens
1-(6-bromo-5-fluoro-1H-indol-3-yl)propan-2-one
-
 Homo sapiens
2-(5,6-dibromo-1H-indol-3-yl)-N-methylethanamine
-
 Homo sapiens
2-(5,6-dibromo-1H-indol-3-yl)ethanamine
-
 Homo sapiens
2-(5,6-dichloro-1H-indol-3-yl)-N-methylethanamine
-
 Homo sapiens
2-(5,6-dichloro-1H-indol-3-yl)ethanamine
-
 Homo sapiens
2-(5,6-difluoro-1H-indol-3-yl)-N-methylethanamine
-
 Homo sapiens
2-(5,6-difluoro-1H-indol-3-yl)ethanamine
-
 Homo sapiens
2-(5-bromo-6-chloro-1H-indol-3-yl)-N-methylethanamine
-
 Homo sapiens
2-(5-bromo-6-chloro-1H-indol-3-yl)ethanamine
-
 Homo sapiens
2-(5-bromo-6-fluoro-1H-indol-3-yl)-N-methylethanamine
-
 Homo sapiens
2-(5-bromo-6-fluoro-1H-indol-3-yl)ethanamine
-
 Homo sapiens
2-(6-bromo-5-chloro-1H-indol-3-yl)-N-methylethanamine
-
 Homo sapiens
2-(6-bromo-5-chloro-1H-indol-3-yl)ethanamine
-
 Homo sapiens
2-(6-bromo-5-fluoro-1H-indol-3-yl)-N-methylethanamine
-
 Homo sapiens
2-(6-bromo-5-fluoro-1H-indol-3-yl)ethanamine
-
 Homo sapiens
5,6-dibromo-3-methyl-1H-indole
-
 Homo sapiens
5,6-dibromo-3-phenyl-1H-indole best inhibitor for glycogen synthetase kinase-3 beta; best inhibitor for glycogen synthetase kinase-3 beta Homo sapiens
5,6-dichloro-3-methyl-1H-indole
-
 Homo sapiens
5,6-dichloro-3-phenyl-1H-indole
-
 Homo sapiens
5,6-difluoro-3-methyl-1H-indole
-
 Homo sapiens
5,6-difluoro-3-phenyl-1H-indole
-
 Homo sapiens
5-bromo-6-chloro-3-methyl-1H-indole
-
 Homo sapiens
5-bromo-6-chloro-3-phenyl-1H-indole
-
 Homo sapiens
5-bromo-6-fluoro-3-methyl-1H-indole
-
 Homo sapiens
5-bromo-6-fluoro-3-phenyl-1H-indole
-
 Homo sapiens
6-bromo-5-chloro-3-methyl-1H-indole
-
 Homo sapiens
6-bromo-5-chloro-3-phenyl-1H-indole
-
 Homo sapiens
6-bromo-5-fluoro-3-methyl-1H-indole
-
 Homo sapiens
6-bromo-5-fluoro-3-phenyl-1H-indole
-
 Homo sapiens
convolutamine I
-
 Homo sapiens
convolutamine J
-
 Homo sapiens
kororamide A
-
 Homo sapiens
kororamide B
-
 Homo sapiens
meridianin F
-
 Homo sapiens

Natural Substrates/ Products (Substrates)

Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
ATP + tau-protein Homo sapiens
-
 ADP + O-phospho-tau-protein
-
 ?

Organism

Organism UniProt Comment Textmining
Homo sapiens P48730
-
-
Homo sapiens P49841
-
-

Source Tissue

Source Tissue Comment Organism Textmining
brain
-
 Homo sapiens
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
ATP + tau-protein
-
 Homo sapiens ADP + O-phospho-tau-protein
-
 ?

Synonyms

Synonyms Comment Organism
casein kinase 1 delta
-
 Homo sapiens
CK1delta
-
 Homo sapiens
glycogen synthetase kinase-3 beta
-
 Homo sapiens
GSK3beta
-
 Homo sapiens
tau protein kinase
-
 Homo sapiens