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Literature summary for 2.7.11.2 extracted from

  • Savkur, R.S.; Bramlett, K.S.; Michael, L.F.; Burris, T.P.
    Regulation of pyruvate dehydrogenase kinase expression by the farnesoid X receptor (2005), Biochem. Biophys. Res. Commun., 329, 391-396.
    View publication on PubMed

Activating Compound

Activating Compound Comment Organism Structure
additional information farnesoid X receptor agonist GW4064 stimulates PDK4 expression in liver in vivo Mus musculus
additional information farnesoid X receptor agonists stimulate PDK4 expression in hepatocytes in vitro Homo sapiens
additional information glucocorticoids and farnesoid X receptor agonists, dexamethasone or WY14643, stimulate PDK4 expression in hepatoma cells in vitro Rattus norvegicus

Natural Substrates/ Products (Substrates)

Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
additional information Mus musculus regulation of pyruvate dehydrogenase kinase expression by the farnesoid X receptor, mechanism ?
-
?
additional information Homo sapiens regulation of pyruvate dehydrogenase kinase expression by the farnesoid X receptor, mechanism ?
-
?
additional information Rattus norvegicus regulation of pyruvate dehydrogenase kinase expression by the farnesoid X receptor, mechanism ?
-
?
additional information Mus musculus C57BL/6 regulation of pyruvate dehydrogenase kinase expression by the farnesoid X receptor, mechanism ?
-
?

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
-
-
Mus musculus
-
C75BL/6 mice
-
Mus musculus C57BL/6
-
C75BL/6 mice
-
Rattus norvegicus
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
H4IIE cell hepatoma cell line, determination of PDK4 expression level in presence or absence of farnesoid X receptor agonists Rattus norvegicus
-
hepatocyte primary, determination of PDK4 expression level in presence or absence of farnesoid X receptor agonists Homo sapiens
-
hepatoma cell
-
Rattus norvegicus
-
liver determination of PDK4 expression level in presence or absence of farnesoid X receptor agonists Mus musculus
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
additional information regulation of pyruvate dehydrogenase kinase expression by the farnesoid X receptor, mechanism Mus musculus ?
-
?
additional information regulation of pyruvate dehydrogenase kinase expression by the farnesoid X receptor, mechanism Homo sapiens ?
-
?
additional information regulation of pyruvate dehydrogenase kinase expression by the farnesoid X receptor, mechanism Rattus norvegicus ?
-
?
additional information regulation of pyruvate dehydrogenase kinase expression by the farnesoid X receptor, mechanism Mus musculus C57BL/6 ?
-
?

Synonyms

Synonyms Comment Organism
PDK4
-
Mus musculus
PDK4
-
Homo sapiens
PDK4
-
Rattus norvegicus
pyruvate dehydrogenase kinase
-
Mus musculus
pyruvate dehydrogenase kinase
-
Homo sapiens
pyruvate dehydrogenase kinase
-
Rattus norvegicus