Any feedback?
Please rate this page
(literature.php)
(0/150)

BRENDA support

Literature summary for 2.7.11.13 extracted from

  • Beltowski, J.; Marciniak, A.; Jamroz-Wisniewska, A.; Borkowska, E.; Wojcicka, G.
    Bidirectional regulation of renal cortical Na+,K+-ATPase by protein kinase C (2004), Acta Biochim. Pol., 51, 757-772.
    View publication on PubMed

Activating Compound

Activating Compound Comment Organism Structure
diacylglycerol
-
Rattus norvegicus
mezerein stimulates classical, but not novel PKC isozymes Rattus norvegicus
phorbol 12,13-dibutyrate activates PKC, activates Na+,K+-ATPase activity at low concentration, but inhibits it at high concentration Rattus norvegicus
phorbol 12-myristate 13-acetate
-
Rattus norvegicus
thymeleatoxin activates Na+,K+-ATPase activity at low concentration, but inhibits it at high concentration Rattus norvegicus

Inhibitors

Inhibitors Comment Organism Structure
GF109203X inhibits classical and novel, but not atypical PKC isozymes Rattus norvegicus
GΓΆ-6976 inhibits classical, but not novel and atypical PKC isozymes Rattus norvegicus
LY333531 specific inhibition of PKCbeta Rattus norvegicus
phorbol 12,13-dibutyrate activates Na+,K+-ATPase activity at low concentration, but inhibits it at high concentration, the inhibitory effect can be reversed by preincubation with ethoxyresorufin, 17-octadecynoic acid, wortmannin, LY294002, cytochlasin D, or latrunculin B Rattus norvegicus
staurosporine inhibits all PKC isozymes Rattus norvegicus
thymeleatoxin activates Na+,K+-ATPase activity at low concentration, but inhibits it at high concentration Rattus norvegicus

Natural Substrates/ Products (Substrates)

Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
additional information Rattus norvegicus bidirectional regulation of renal cortical Na+,K+-ATPase by PKC ?
-
?

Organism

Organism UniProt Comment Textmining
Rattus norvegicus
-
male Wistar rats
-

Source Tissue

Source Tissue Comment Organism Textmining
kidney
-
Rattus norvegicus
-
renal cortex
-
Rattus norvegicus
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
additional information bidirectional regulation of renal cortical Na+,K+-ATPase by PKC Rattus norvegicus ?
-
?

Synonyms

Synonyms Comment Organism
PKC
-
Rattus norvegicus