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Literature summary for 2.7.11.11 extracted from

  • Komalavilas, P.; Penn, R.B.; Flynn, C.R.; Thresher, J.; Lopes, L.B.; Furnish, E.J.; Guo, M.; Pallero, M.A.; Murphy-Ullrich, J.E.; Brophy, C.M.
    The small heat shock-related protein, HSP20, is a cAMP-dependent protein kinase substrate that is involved in airway smooth muscle relaxation (2008), Am. J. Physiol. Lung Cell Mol. Physiol., 294, L69-L78.
    View publication on PubMedView publication on EuropePMC

Activating Compound

Activating Compound Comment Organism Structure
forskolin activation at 0.01 mM Bos taurus
isoproterenol activation at 0.001 mM Bos taurus

Inhibitors

Inhibitors Comment Organism Structure
PKI
-
Bos taurus

Organism

Organism UniProt Comment Textmining
Bos taurus
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
airway smooth muscle
-
Bos taurus
-
airway smooth muscle cell
-
Bos taurus
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
ATP + small heat shock-related protein HSP20
-
Bos taurus ADP + phosphorylated small heat shock-related protein HSP20
-
?

Synonyms

Synonyms Comment Organism
PKA
-
Bos taurus
protein kinase A
-
Bos taurus

Cofactor

Cofactor Comment Organism Structure
ATP
-
Bos taurus
cAMP dependent Bos taurus