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Literature summary for 2.7.10.2 extracted from

  • Huang, Y.; Comiskey, E.O.; Dupree, R.S.; Li, S.; Koleske, A.J.; Burkhardt, J.K.
    The c-Abl tyrosine kinase regulates actin remodeling at the immune synapse (2008), Blood, 112, 111-119.
    View publication on PubMedView publication on EuropePMC

Inhibitors

Inhibitors Comment Organism Structure
imatinib mesylate
-
Homo sapiens

Natural Substrates/ Products (Substrates)

Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
ATP + [protein]-L-tyrosine Homo sapiens
-
ADP + [protein]-L-tyrosine phosphate
-
?

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
JURKAT cell JURKAT T cell Homo sapiens
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
ATP + [actin-stabilizing adapter protein HS1]-L-tyrosine c-Abl binds to phospho-HS1 via its SH2 domains and is required for full tyrosine phosphorylation of HS1 during T-cell activation Homo sapiens ADP + [actin-stabilizing adapter protein HS1]-L-tyrosine phosphate
-
?
ATP + [protein]-L-tyrosine
-
Homo sapiens ADP + [protein]-L-tyrosine phosphate
-
?

Synonyms

Synonyms Comment Organism
c-Abl tyrosine kinase
-
Homo sapiens

Temperature Optimum [°C]

Temperature Optimum [°C] Temperature Optimum Maximum [°C] Comment Organism
30
-
in vitro kinase assay Homo sapiens

pH Optimum

pH Optimum Minimum pH Optimum Maximum Comment Organism
7.2
-
in vitro kinase assay Homo sapiens

Cofactor

Cofactor Comment Organism Structure
ATP
-
Homo sapiens