Inhibitors | Comment | Organism | Structure |
---|---|---|---|
1,4-diamino-2,3-dicyano-1,4-bis(2-aminophenylthio)-butadiene | - |
Homo sapiens | |
afatinib | - |
Homo sapiens | |
BI2536 | - |
Homo sapiens | |
canertinib | - |
Homo sapiens | |
crizotinib | - |
Homo sapiens | |
dacomitinib | - |
Homo sapiens | |
dasatinib | - |
Homo sapiens | |
erlotinib | - |
Homo sapiens | |
gefitinib | - |
Homo sapiens | |
imatinib | - |
Homo sapiens | |
KU55933 | - |
Homo sapiens | |
lapatinib | dual inhibitor of EGFR and ERBB2 | Homo sapiens | |
LY2874455 | - |
Homo sapiens | |
neratinib | - |
Homo sapiens | |
NVP-BEZ235 | - |
Homo sapiens | |
PD184352 | - |
Homo sapiens | |
PD325901 | - |
Homo sapiens | |
PD98059 | - |
Homo sapiens | |
PIK-90 | - |
Homo sapiens | |
PI_103 | - |
Homo sapiens | |
sorafenib | - |
Homo sapiens | |
staurosporine | - |
Homo sapiens | |
trastuzumab | - |
Homo sapiens | |
tyrphostin | - |
Homo sapiens | |
varlitinib | - |
Homo sapiens | |
ZSTK474 | - |
Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
- |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
BT474 cell | - |
Homo sapiens | - |
BT474-LR cell | - |
Homo sapiens | - |
Synonyms | Comment | Organism |
---|---|---|
Egfr | - |
Homo sapiens |
ErbB2 | - |
Homo sapiens |
ErbB4 | - |
Homo sapiens |
HER2 | - |
Homo sapiens |
HER4 | - |
Homo sapiens |
General Information | Comment | Organism |
---|---|---|
physiological function | ERBB4 plays a key role in the survival of ERBB2C cancer cells after they develop resistance to ERBB2 inhibitors, lapatinib and trastuzumab | Homo sapiens |