Activating Compound | Comment | Organism | Structure |
---|---|---|---|
D-fructose 1,6-bisphosphate | activates | Homo sapiens |
Application | Comment | Organism |
---|---|---|
diagnostics | its presence in human plasma is currently being used as a molecular marker for the diagnosis of various cancers | Homo sapiens |
Crystallization (Comment) | Organism |
---|---|
the X-ray structure of human hPKM2 complexed with Mg2+, K+, the inhibitor oxalate, and the allosteric activator D-fructose 1,6-bisphosphate determined to a resolution of 2.82 A. (His)6-tagged hPKM2 complex, hanging drop vapor diffusion | Homo sapiens |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.17 | - |
phosphoenolpyruvate | pH 8.0, 32°C, activation by 2 mM D-fructose-1,6-bisphosphate | Homo sapiens | |
0.24 | - |
ADP | pH 8.0, 32°C, activation by 2 mM D-fructose-1,6-bisphosphate | Homo sapiens | |
0.34 | - |
ADP | pH 8.0, 32°C | Homo sapiens | |
2.1 | - |
phosphoenolpyruvate | pH 8.0, 32°C | Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | P14618 | - |
- |
Purification (Comment) | Organism |
---|---|
- |
Homo sapiens |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
blood plasma | - |
Homo sapiens | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
ADP + phosphoenolpyruvate | - |
Homo sapiens | ATP + pyruvate | - |
? |
Synonyms | Comment | Organism |
---|---|---|
hPKM2 | pyruvate kinase isoenzyme M2 | Homo sapiens |