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Literature summary for 2.7.1.137 extracted from

  • Linassier, C.; MacDougall, L.K.; Domin, J.; Waterfield, M.D.
    Molecular cloning and biochemical characterization of a Drosophila phosphatidylinositol-specific phosphoinositide 3-kinase (1997), Biochem. J., 321, 849-856.
No PubMed abstract available

Cloned(Commentary)

Cloned (Comment) Organism
expression of the complete coding sequence as a glutathione S-transferase fusion protein in Sf9 cells Drosophila melanogaster

Inhibitors

Inhibitors Comment Organism Structure
Nonidet P40
-
Drosophila melanogaster
Wortmannin IC50 10 nM Drosophila melanogaster

Organism

Organism UniProt Comment Textmining
Drosophila melanogaster P91635
-
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
ATP + 1-phosphatidylinositol
-
Drosophila melanogaster ADP + phosphatidylinositol 3-phosphate
-
?

Synonyms

Synonyms Comment Organism
PI3K_59F
-
Drosophila melanogaster

IC50 Value

IC50 Value IC50 Value Maximum Comment Organism Inhibitor Structure
0.00001
-
IC50 10 nM Drosophila melanogaster Wortmannin