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Literature summary for 2.7.1.137 extracted from

  • Sato, M.; Bryant, H.U.; Dodge, J.A.; Davis, H.; Matter, W.F.; Vlahos, C.J.
    Effects of wortmannin analogs on bone in vitro and in vivo (1996), J. Pharmacol. Exp. Ther., 277, 543-550.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
LY301497
-
Bos taurus
LY301497
-
Gallus gallus
Wortmannin
-
Bos taurus
Wortmannin
-
Gallus gallus
Wortmannin
-
Rattus norvegicus

Natural Substrates/ Products (Substrates)

Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
additional information Gallus gallus PI 3-kinase activity is a necessary step in the regulation of bone resorption ?
-
?
additional information Bos taurus PI 3-kinase activity is a necessary step in the regulation of bone resorption ?
-
?
additional information Rattus norvegicus PI 3-kinase activity appears to be an important component of ovariectomy-stimulated bone loss in rats ?
-
?

Organism

Organism UniProt Comment Textmining
Bos taurus
-
-
-
Gallus gallus
-
-
-
Rattus norvegicus
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
osteoclast
-
Gallus gallus
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
ATP + 1-phosphatidylinositol
-
Gallus gallus ADP + phosphatidylinositol 3-phosphate
-
?
ATP + 1-phosphatidylinositol
-
Rattus norvegicus ADP + phosphatidylinositol 3-phosphate
-
?
ATP + 1-phosphatidylinositol
-
Bos taurus ADP + phosphatidylinositol 3-phosphate
-
?
additional information PI 3-kinase activity is a necessary step in the regulation of bone resorption Gallus gallus ?
-
?
additional information PI 3-kinase activity is a necessary step in the regulation of bone resorption Bos taurus ?
-
?
additional information PI 3-kinase activity appears to be an important component of ovariectomy-stimulated bone loss in rats Rattus norvegicus ?
-
?