Activating Compound | Comment | Organism | Structure |
---|---|---|---|
deoxycholate | stimulation | Catharanthus roseus | |
phosphatidylglycerol | effective stimulation | Catharanthus roseus | |
phosphatidylinositol | effective stimulation | Catharanthus roseus |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
ADP | - |
Catharanthus roseus | |
ATP | - |
Catharanthus roseus | |
ATPgammaS | - |
Catharanthus roseus | |
CDP | - |
Catharanthus roseus | |
CTP | - |
Catharanthus roseus | |
GDP | - |
Catharanthus roseus | |
GDPbetaS | - |
Catharanthus roseus | |
GTP | - |
Catharanthus roseus | |
IDP | - |
Catharanthus roseus | |
ITP | - |
Catharanthus roseus | |
phosphate | - |
Catharanthus roseus | |
UDP | - |
Catharanthus roseus | |
UTP | - |
Catharanthus roseus |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
additional information | - |
additional information | in presence of Triton X-100, used for purification, a biphasic dependency upon diacylglycerol is observed and the apparent Michaelis constant values for diacylglycerol decreases with decreasing Triton concentration | Catharanthus roseus | |
0.102 | - |
ATP | pH 7.5, 25°C | Catharanthus roseus | |
0.104 | - |
GTP | pH 7.5, 25°C | Catharanthus roseus | |
0.9 | - |
dioleoylglycerol | pH 7.5, 25°C | Catharanthus roseus |
Localization | Comment | Organism | GeneOntology No. | Textmining |
---|---|---|---|---|
cytosol | no activity in cytosol | Catharanthus roseus | 5829 | - |
membrane | intrinsic membrane-protein | Catharanthus roseus | 16020 | - |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Catharanthus roseus | - |
- |
- |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
ATP + sn-1,2-dioleoylglycerol | - |
Catharanthus roseus | ADP + sn-1,2-dioleoylglycerol 3-phosphate | - |
? | |
GTP + dioleoylglycerol | - |
Catharanthus roseus | GDP + dioleoylglycerol 3-phosphate | - |
? |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.038 | - |
IDP | pH 7.5, 25°C | Catharanthus roseus | |
0.043 | - |
UDP | pH 7.5, 25°C | Catharanthus roseus | |
0.058 | - |
GDP | pH 7.5, 25°C | Catharanthus roseus | |
0.06 | - |
CDP | pH 7.5, 25°C | Catharanthus roseus | |
0.081 | - |
GTP | pH 7.5, 25°C | Catharanthus roseus | |
0.095 | - |
ADP | pH 7.5, 25°C | Catharanthus roseus | |
0.102 | - |
ATP | pH 7.5, 25°C | Catharanthus roseus | |
0.123 | - |
GDPbetaS | pH 7.5, 25°C | Catharanthus roseus | |
0.26 | - |
UTP | pH 7.5, 25°C | Catharanthus roseus | |
0.48 | - |
CTP | pH 7.5, 25°C | Catharanthus roseus | |
0.51 | - |
ITP | pH 7.5, 25°C | Catharanthus roseus | |
2.5 | - |
phosphate | pH 7.5, 25°C | Catharanthus roseus |