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Literature summary for 2.3.1.87 extracted from

  • Tsuboi, S.; Kotani, Y.; Ogawa, K.i.; Hatanaka, T.; Yatsushiro, S.; Otsuka, M.; Moriyama, Y.
    An Intramolecular Disulfide Bridge as a Catalytic Switch for Serotonin N-Acetyltransferase (2002), J. Biol. Chem., 277, 44229-44235.
    View publication on PubMed

Protein Variants

Protein Variants Comment Organism
C177A fully active, not sensitive to oxidation or N-ethylmaleimide Rattus norvegicus
C61A fully active, not sensitive to oxidation or N-ethylmaleimide Rattus norvegicus

Inhibitors

Inhibitors Comment Organism Structure
glutathione reversible, acetyl-CoA protects Rattus norvegicus
N-ethylmaleimide irreversible, acetyl-CoA protects Rattus norvegicus
oxygen reversible, acetyl-CoA protects Rattus norvegicus

KM Value [mM]

KM Value [mM] KM Value Maximum [mM] Substrate Comment Organism Structure
additional information
-
additional information formation and cleavage of a disulfide bond produce active/inactive states of enzyme Rattus norvegicus

Organism

Organism UniProt Comment Textmining
Rattus norvegicus Q64666
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