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Literature summary for 1.5.1.33 extracted from

  • Kaur, J.; Singh, N.; Singh, B.K.; Dube, A.; Tripathi, R.P.; Singh, P.; Singh, N.
    Leishmania donovani: oral therapy with glycosyl 1,4-dihydropyridine analogue showing apoptosis like phenotypes targeting pteridine reductase 1 in intracellular amastigotes (2010), Exp. Parasitol., 125, 310-314.
    View publication on PubMed

Cloned(Commentary)

Cloned (Comment) Organism
transgenic parasites overexpress a PTR1-GFP chimera (PTR1 tagged at the N-terminal with GFP) Leishmania major

Inhibitors

Inhibitors Comment Organism Structure
2,6-dimethyl-4-(3-O-benzyl-1,2-O-isopropylidene-beta-L-threo pentofuranos-4-yl)-1-phenyl-1,4-dihydro-pyridine-3,5-dicarboxylic acid diethyl ester oral therapy shows apoptosis like phenotypes targeting pteridine reductase 1 in intracellular amastigotes Leishmania major

Localization

Localization Comment Organism GeneOntology No. Textmining

Organism

Organism UniProt Comment Textmining
Leishmania major
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining

Synonyms

Synonyms Comment Organism
pteridine reductase 1
-
Leishmania major
PTR1
-
Leishmania major