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Literature summary for 1.1.1.205 extracted from

  • Yamada, Y.; Goto, H.; Yoshino, M.; Ogasawara, N.
    IMP dehydrogenase and action of antimetabolites in human cultured blast cells (1990), Biochim. Biophys. Acta, 1051, 209-214.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
NADH
-
Homo sapiens
ribavirin 5'-monophosphate competitive with respect to IMP Homo sapiens
thiazole-4-carboxamide adenine dinucleotide inhibitory mechanism Homo sapiens
tiazofurin
-
Homo sapiens
xanthosine 5'-phosphate
-
Homo sapiens

KM Value [mM]

KM Value [mM] KM Value Maximum [mM] Substrate Comment Organism Structure
additional information
-
additional information
-
Homo sapiens

Molecular Weight [Da]

Molecular Weight [Da] Molecular Weight Maximum [Da] Comment Organism
60000
-
SDS-PAGE Homo sapiens

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
-
-

Purification (Commentary)

Purification (Comment) Organism
MOLT 4F human T-lymphoblasts Homo sapiens

Source Tissue

Source Tissue Comment Organism Textmining
B-lymphoblast
-
Homo sapiens
-
BALL-1 cell
-
Homo sapiens
-
K-562 cell
-
Homo sapiens
-
MOLT-4F cell
-
Homo sapiens
-

Specific Activity [micromol/min/mg]

Specific Activity Minimum [µmol/min/mg] Specific Activity Maximum [µmol/min/mg] Comment Organism
additional information
-
-
Homo sapiens

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
inosine 5'-phosphate + NAD+ + H2O
-
Homo sapiens xanthosine 5'-phosphate + NADH
-
?

Cofactor

Cofactor Comment Organism Structure
NAD+
-
Homo sapiens

Ki Value [mM]

Ki Value [mM] Ki Value maximum [mM] Inhibitor Comment Organism Structure
0.000075
-
thiazole-4-carboxamide adenine dinucleotide
-
Homo sapiens
0.00058
-
ribavirin 5'-monophosphate
-
Homo sapiens
0.085
-
xanthosine 5'-phosphate
-
Homo sapiens
0.094
-
NADH
-
Homo sapiens